Inquire About a ProductActivators
An Activator is a substance that increases the effectiveness of another. For example, a trace quantity of a substance that imparts luminescence to crystals; silver or copper in zinc sulfide or cadmium sulfide pigments. In genetics it would be a molecule that modifies a repressor in a way that enables it to stimulate operon transcription. Examples of activators are: 1-Acetamido-4-cyano-3-methylisoquinoline that is used as a selective inhibitor of cyclic AMP-dependent protein kinase (PKA), while D-erythro-Dihydro-D-sphingosine is used as a Biosynthetic precursor of sphingosine, Inhibits protein kinase C.
Chemical Activators
Protein Kinase Inhibitors and Activators
| Catalog No. | Product Name | Enrichment |
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| 18445 |
Acitazanolast
Synonyms: 2-(3-(1H-tetrazol-5-yl)phenylamino)-2-oxoacetic acid; |
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| 6411 |
N-(4-Aminobutyl)-2-naphthalenesulfonamide HCl
Synonyms: W-12; |
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| 6467 | N-(10-Aminodecyl)-5-chloro-1-naphthalenesulfonamide HCl |
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| 6546 |
N-(2-Aminoethyl)-5-chloro-1-naphthalenesulfonamide HCl
Synonyms: A-3; |
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| 6582 |
N-(6-Aminohexyl)-1-naphthalenesulfonamide HCl
Synonyms: W-5; |
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| 7731 | N-[2-(p-Bromocinnamylamino)ethyl]-5-Isoquinoline Sulfonamide |
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| 7732 | N-[2-(p-Bromocinnamylamino)ethyl]-5-isoquinoline Sulfonamide DiHCl |
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| D17294 |
Bromoenol lactone-d7
Synonyms: (S)-BEL-d7; 6E-(bromoethylene)tetrahydro-3S-(1-naphthalenyl-2,3, 4,5,6,7,8-d7)-2H-pyran-2-one; |
99% D |
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| 7454 | 1,3-Bis-(o-tert-butyldimethylsilyl)-Fmoc-D-erythro-sphingosine |
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| 8213 |
C22 Ceramide
Synonyms: N-[(3E)-2-hydroxy-1-(hydroxymethyl)-3-heptadecenyl]-docosanamide; |
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| 8214 |
C22 Dihydroceramide
Synonyms: N-[(1S,2R)-2-Hydroxy-1-(hydroxymethyl)-heptadecyl]-docosanamide; |
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| 8349 |
1-(8-Chloro-5-isoquinolinesulfonyl)piperazine DiHCl
Synonyms: HA-156; |
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| 8503 |
N-[2-(p-Cinnamylamino)ethyl]-5-isoquinolone Sulfonamide
Synonyms: H-88; |
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| D2670 | Daidzein-d4 | 92%D |
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| 32095 |
N,N-Dimethylsphingosine
Synonyms: 2-Dimethylamino-4-octadecene-1,3-diol; D-erythro-N,N-Dimethylsphingosine; |
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| 94009 |
rac-1,2-Dipalmitoylglycerol
Synonyms: Hexadecanoic Acid 1-(Hydroxymethyl)-1,2-ethanediyl Ester; (±)- Hexadecanoic Acid 1-(Hydroxymethyl)-1,2-ethanediyl Ester; (RS)-1, 2-Dipalmitin; (±)-1,2-Dipalmitin; (±)-1,2-Dipalmitoylglycerin; (±)-1,2-Dipalmitoylglycerol; (±)-1-(Hydroxymethyl)ethane-1,2- diyl dipalmitate; 1,2-Dipalmitin; 1,2-Dipalmitoyl-DL-glycerol; 1, 2-Dipalmitoyl-rac-glycerol; 1,2-Dipalmitoylglycerol; 2,3- Dipalmitin; Glycerol 1,2-dihexadecanoate; Glycerol 1,2- dipalmitate; rac-Glycerol 1,2-dipalmitate; |
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| 9485 |
D-erythro-Dihydro-D-sphingosine
Synonyms: Sphinganine; |
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| 9486 | D-erythro-Dihydro-D-sphingosine-1-phosphate |
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| D32096 | D-erythro-N,N-Dimethylsphingosine-d6 |
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| 18625 |
Fasudil HCl
Synonyms: 5-(1,4-diazepane-1-sulfonyl)isoquinoline; |
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| 10606 |
N-(N-Heptyl)-5-chloro-1-naphthalenesulfonamide
Synonyms: SC-10; |
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| 11077 |
10Z-Hymenialdisine
Synonyms: 4-(2-Amino-4-oxo-2-imidazolidin-5-ylidene)-2-bromo-4,5,6,7- tetrahydropyrrolo[2,3-c]azepin-8-one; |
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| 11078 |
Hymenialdisine Analogue #1
Synonyms: 5-(2-Amino-5-oxo-1,5-dihydroimidazol-4-ylidene)-3,4,5,10- tetrahydro-2H-azepino[3,4-β]indol-1-one; |
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| 11238 |
1-(5-Isoquinolinesulfonyl)-1H-hexahydro-1,4-diazepine DiHCl
Synonyms: HA1077 Dihydrochloride; Fasudildihydrochloride; 1-(5-Isoquinolinylsulfonyl)homopiperazinedihydrochloride; |
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| 71002 | 1-(5-Isoquinolinesulfonyl)-2-methyl-4-trityl-piperazine |
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| 71001 | 1-(5-Isoquinolinesulfonyl)-4-tert-butyloxycarbonyl-2- methylpiperazine |
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| 11242 |
1-(5-Isoquinolinesulfonyl)piperazine DiHCl
Synonyms: HA-100 dihydrochloride; 1-(5-Isoquinolinesulfonyl)piperazine dihydrochloride; |
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| 11303 |
KN-62
Synonyms: (S)-5-Isoquinolinesulfonic acid 4-[2-[(5-isoquinolinylsulfonyl) methylamino]-3-oxo-3-(4-phenyl-1-piperazinyl)propyl]phenyl ester; 1-[N,O-bis(5-Isoquinolinesulfonyl)-N-methyl-L-tyrosyl]-4- phenylpiperazine; |
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| 11776 |
N-[2-(Methylamino)ethyl]-5-isoquinolinesulfonamide DiHCl
Synonyms: H-8; N-[2-(Methylamino)ethyl]-5-isoquinolinesulfonamidehydrochloride; |
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| D97819 | Nonadecanoic Acid 3-(Acetyloxy)-2-hydroxypropyl Ester-d5 |
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| 13045 |
N-(6-Phenylhexyl)-5-chloro-1-naphthalenesulfonamide
Synonyms: SC-9; |
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| 14868 |
SNS-032
Synonyms: BMS-387032; BMS-387072; CID3025986; LS-186036; N-(5-(((5-(1,1-Dimethylethyl)-2-oxazolyl)methyl)thio)-2-thiazolyl )-4-piperidinecarboxamide; 4-Piperidinecarboxamide; N-(5-(((5-(1,1-dimethylethyl)-2-oxazolyl)methyl)thio)-2-thiazolyl )-; N-[5-[(5-tert-butyl-1,3-oxazol-2-yl)methylsulfanyl]-1,3-thiazol-2 -yl]piperidine-4-carboxamide; |
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| 13631 |
Tamoxifen
Synonyms: (Z)-2-[4-(1,2-Diphenyl-1-butenyl)phenoxy]-N,N-dimethylethanamine; Trans-2-[4-(1,2-Diphenyl-1-butenyl)phenoxy]-N,N- dimethylethylamine; |
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| 14848 |
Telaprevir
Synonyms: (1S,3aR,6aS)-2-[(2S)-2-[[(2S)-2-Cyclohexyl-2-(pyrazine-2- carbonylamino)acetyl]amino]-3,3-dimethylbutanoyl]-N-[(3S)-1- (cyclopropylamino)-1,2-dioxohexan-3-yl]-3,3a,4,5,6,6a-hexahydro- 1H-cyclopenta[c]pyrrole-1-carboxamide; VX-950; |
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| 13706 |
4,5,6,7-Tetrabromo-1H-benzotriazole
Synonyms: TBB; 4,5,6,7-Tetrabromo-2-azabenzimidazole; 4,5,6,7-Tetrabromobenzotriazole; NSC 231634; TBBt; |
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| 13705 |
4,5,6,7-Tetrabromobenzimidazole
Synonyms: TBBz; |
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| 18796 | Trapidil |
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| 14033 |
3,4,5-Trimethoxybenzoic Acid 8-(Diethylamino)octyl Ester HCl
Synonyms: TMB-8 HCl; |
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| D99882 |
Trimyristin-d5
Synonyms: Tetradecanoic Acid 1,1’,1’’-(1,2,3-propanetriyl) Ester-d5; Dynasan 114-d5; Glycerin Trimyristate-d5; Glycerol Trimyristate- d5; Glyceryl Trimyristate-d5; Glyceryl Tritetradecanoate-d5; Myristic Acid Triglyceride-d5; Myristic Triglyceride-d5; NSC 4062 -d5; Triglyceride MMM-d5; Trimyristin-d5; Trimyristoylglycerol- d5; Tritetradecanoin-d5; VP 114-d5; |
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| 14615 | Vatalanib base |
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| 14616 |
Vatalanib succinate
Synonyms: N-(4-Chlorophenyl)-4-(4-pyridinylmethyl)-1-phthalazinamine butanedioate; |
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Agonists
| Catalog No. | Product Name | Enrichment |
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|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 38386 | A 61603 |
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| 18438 |
Abecarnil
Synonyms: 6-(Benzyloxy)-4-(methoxymethyl)-β-carboline-3-carboxylic acid isopropyl ester; |
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| 18442 | Aceclidine |
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| D38429 | 4-Acetamido-5-chloro-2-ethoxy-benzoic Acid Methyl Ester-d5 |
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| D19066 |
4-Acetamido-5-chloro-2-ethoxybenzoic Acid Methyl Ester-d5
Synonyms: Methyl 4-acetamido-5-chloro-2-ethoxybenzoate-d5; |
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| D312 |
Acetylcholine-d9 Bromide
Synonyms: (2-Acetoxyethyl)trimethylammonium-d9 Bromide; 2-(Acetyloxy)-N,N,N-trimethylethanaminium-d9 Bromide; |
99%D |
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| D315 | Acetylcholine-1,1,2,2-d4 Chloride | 99%D |
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| D4878 |
Acetylcholine-d9 Chloride
Synonyms: (2-Acetoxyethyl)trimethylammonium-d9 Chloride; |
99%D |
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| 18446 | Aclatonium Napadisilate |
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| C19360 |
Adenosine-13C5
Synonyms: 9-β-D-Ribofuranosyl-9H-purin-6-amine-13C5; 9-β-D-Ribofuranosyladenine-13C5; Adenine Riboside-13C5; Adenocard-13C5; Adenocor-13C5; Adenogesic-13C5; Adenoscan-13C5; Adrekar-13C5; Boniton-13C5; D-Adenosine-13C5; 1-(6-Amino-9H-purin-9-yl)-1-deoxy-β-D; |
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| 38491 | AdipoRon |
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| 38497 | AH 7921 HCl |
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| 5714 |
Albuterol
Synonyms: Salbutamol; |
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| D4526 |
Albuterol-d9
Synonyms: a1-[[(1,1-Dimethylethyl)amino]methyl]-4-hydroxy-1,3- benzenedimethanol-d9; Salbutamol-d9; |
98%D |
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| D74808 | Albuterol-d3 |
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| 38512 | Alda 1 |
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| 18461 | Aleglitazar |
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| 38529 | 6-Allyl-8β-carboxyergoline Methyl Ester |
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| 18470 |
Almitrine
Synonyms: 6-[4-[bis(4-fluorophenyl)methyl]piperazin-1-yl]-N,N’-diprop-2- enyl-1,3,5-triazine-2,4-diamine; |
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| D6315 |
Almotriptan-d6 Hydrochloride
Synonyms: 1-[[[2-(Dimethyl-amino)ethyl]-1H-indol-5-yl]methyl]sulfonyl] pyrrolidine-d6; 1-[[3-(2-dimethylaminoethyl)-5-indolyl]methanesulfonyl] pyrrolidine-d6; LAS-31416-d6; |
98%D |
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| 38541 | AM-694 |
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| D38542 | AM-694-d4 |
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| 38623 | 3’-Amino-2’-Hydroxy-[1,1’]biphenyl-3-carboxylic Acid |
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| 38621 | 3-Amino-4-hydroxybenzeneacetic Acid |
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| D19603 |
4-Amino-5-chloro-2-ethoxybenzoic Acid-d5
Synonyms: 2-Ethoxy-4-amino-5-chlorobenzoic Acid-d5; |
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| 38725 | (-)-Anatoxin A |
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| 38737 | Arachidonyl-2-chloroethylamide |
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| 18506 | Azepexole |
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| C5342 |
Baclofen-13C2
Synonyms: (RS)-4-amino-3-(4-chlorophenyl)butanoic acid; |
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| 38834 | 2-(Benzofuran-2-yl)-2-imidazoline HCl |
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| D38835 | 2-(Benzofuran-2-yl)-2-imidazoline-d4 HCl |
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| 38906 | (E)-1,2-Bis(1-benzyl-1H-imidazol-5-yl)ethene |
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| 38845 | 3-Benzyl-3H-imidazole-4-carboxaldehyde |
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| 38846 | (E)-1-Benzyl-5-((6-methoxy-2,3-dihydro-1H-inden-1-ylidene)methyl) -1H-imidazole |
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| 38856 | 3-(Benzyloxy)-4-methoxyphenylacetic Acid |
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| D38892 | Betulin-d3 |
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| D38893 | Betulinic Acid-d3 |
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| 38944 | Bisphenol F |
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| D38945 | Bisphenol F-d10 |
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| N38979 | 1N-Boc-6-cyano-6-norlysergol |
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| 18530 |
Brimonidine
Synonyms: 5-Bromo-N-(4,5-dihydro-1H-imidazol-2-yl)-6-quinoxalinamine; 5-Bromo-6-(2-imidazolin-2-ylamino)quinoxaline; Bromoxidine; AGN-190342; UK-14304; |
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| 7690 |
Brimonidine D-Tartrate
Synonyms: 5-Bromo-N-(4,5-dihydro-1H-imidazol-2-yl)-6-quinoxalinamine D- Tartrate; 5-Bromo-6-(2-imidazolin-2-ylamino)quinoxaline; UK-14304-18; AGN-190342-LF; A lphagan; |
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| D18872 |
Brimonidine-d4 L-Tartrate
Synonyms: 5-Bromo-N-(4,5-dihydro-1H-imidazol-d4-2-yl)-6-quinoxalinamine L- Tartrate; 5-Bromo-6-(2-imidazolin-d4-2-ylamino)quinoxaline L-Tartrate; UK-14304-18-d4; AGN-190342-LF-d4; A lphagan-d4; |
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| D7689 |
Brimonidine-d4
Synonyms: 5-Bromo-N-(4,5-dihydro-1H-imidazol-d4-2-yl)-6-quinoxalinamine; 5-Bromo-6-(2-imidazolin-d4-2-ylamino)quinoxaline; Bromoxidine-d4; AGN-190342-d4; UK-14304-d4; |
98%D |
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| D7691 |
Brimonidine-d4 D-tartrate
Synonyms: 5-Bromo-N-(4,5-dihydro-1H-imidazol-d4-2-yl)-6-quinoxalinamine D-Tartrate; 5-Bromo-6-(2-imidazolin-d4-2-ylamino)quinoxaline; UK-14304-18-d4; AGN-190342-LF-d4; A lphagan-d4; |
98%D |
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| 7778 | 2-Bromomelatonin |
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| 39129 | Broxaterol |
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| D39130 | Broxaterol-d9 |
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| 39217 | BzATP Ethylammonium Salt |
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| 8132 |
Cardiogenol C HCl
Synonyms: 4-(2-Hydroxyethylamino)-2-(4-methoxyphenylamino)- pyrimidinehydrochloride; |
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| D39258 | Cardiogenol C-d4, HCl |
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| 39464 | Cinitapride Tartrate |
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| 8510 |
Cisapride
Synonyms: cis-4-Amino-5-chloro-N-[1-([3-(4-fluorophenoxy)propyl]-3-methoxy- 4-piperidinyl]-2-methoxybenzamide; |
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| D8511 |
Cisapride-d3
Synonyms: cis-4-Amino-5-chloro-N-[1-([3-(4-fluorophenoxy)propyl]-3-methoxy- d3-4-piperidinyl]-2-methoxybenzamide; |
98%D |
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| 39477 | CL 316243 Disodium Salt |
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| 22554 |
CP-135807
Synonyms: 3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-N-(3-nitro-2-pyridinyl)- 1H-indol-5-amine; (R)-3-[(1-Methyl-2-pyrrolidinyl)methyl]-N-(3-nitro-2-pyridinyl)- 1H-indol-5-amine; |
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| 39503 | CP-775146 |
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| 39548 | 4-Cyclohexyl-4-(hydroxymethyl)-N-(tert-butoxycarbonyl)piperidine |
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| 39645 | Defluoro Hydroxy AM-694 |
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| D39646 | Defluoro Hydroxy AM-694-d4 |
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| 39647 | Defluoro Tosyloxy AM-694 |
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| D39648 | Defluoro Tosyloxy AM-694-d4 |
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| 39849 | (8β)-9,10-Didehydro-8-[[[(1,1-dimethylethyl)dimethylsilyl] oxy]methyl]-6-methylergoline |
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| D39956 | Dihydro Cabergoline-(d5 major) |
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| 39958 | trans-Dihydro Lisuride |
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