Drug Analogues

A survey of novel small-molecule therapeutics reveals that the majority of them result from analogue design and that their market value represents two-thirds of all small-molecule sales. In natural science, the term analogue, derived from the Latin and Greek analogia, has always been used to describe structural and functional similarity. Extended to drugs, this definition implies that the analogue of an existing drug molecule shares structural and pharmacological similarities with the original compound. Formally, this definition allows the establishment of three categories of drug analogues: analogues possessing chemical and pharmacological similarities (direct analogues); analogues possessing structural similarities only (structural analogues); and chemically different compounds displaying similar pharmacological properties (functional analogues).

Drug Analogues Alphabetic Listing

Catalog No. Product Name Enrichment
Quantity Price
19885 Amino Tadalafil
Synonyms:
(6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a- hexahydropyrazino[1’,2’:1,6]pyrido[3,4-b]indole-1,4-dione;
2.5 mg $890   Add to Cart
25 mg $2,620   Add to Cart
18046 21-Aminoepothilone B
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6743 D-threo-1-(4-Aminophenyl)-2-dichloroacetylamino-1,3-propanediol HCl
100 mg $875   Add to Cart
0.5 g $2,000   Add to Cart
6829 Amisulpride
Synonyms:
4-Amino-N-[(1-ethyl-2-pyrrolidinyl)methyl]-5-(ethylsulfonyl)-2- methoxybenzamide; Aminosultopride; DAN-2163; Socian; Solian; Sulamid;
1 g $495   Add to Cart
D74204 Amisulpride-d5
10 mg $1,900   Add to Cart
25 mg $400   Add to Cart
63064 rac 4-Azido Deprenyl
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7005 4-Azidodeprenyl
Synonyms:
4-Azido-Selegiline;
5 mg $840   Add to Cart
25 mg $1,720   Add to Cart
7747 trans-(E)-1-Bromo-2-[4-[2-(dimethylamino)ethoxy]phenyl]-1,2- diphenylethene
10 mg $830   Add to Cart
50 mg $1,640   Add to Cart
7748 (E,Z)-1-Bromo-2-[4-[2-(dimethylamino)ethoxy]phenyl]-1,2- diphenylethene
25 mg $830   Add to Cart
125 mg $1,640   Add to Cart
8448 D-threo-1-(4-Chlorosulfonylphenyl)-2-dichloroacetylamino-1,3- propanediol
25 mg $860   Add to Cart
125 mg $1,880   Add to Cart
63757 CK 1827452
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D63758 CK 1827452-d8
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63906 DAMPA
50 mg $650   Add to Cart
500 mg $2,200   Add to Cart
D63907 DAMPA-d3
2.5 mg $650   Add to Cart
25 mg $2,200   Add to Cart
CD63991 9,11-Dehydro-17α-cyanomethyl Estradiol-13C,d2
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8811 Demethylchlorocitalopram
1 mg $860   Add to Cart
5 mg $1,880   Add to Cart
8827 Deoxy Artemisinin
Synonyms:
(3R,3aS,6R,6aS,9S,10aS,10bR)-Octahydro-3,6,9-trimethyl-10aH-9,10b -epoxypyrano[4,3,2-jk][2]benzoxepin-2(3H)-one; Deoxyarteannuin; Deoxyartemisinin; Deoxyqinghaosu; Desoxyartemisinin; Hydroarteannuin; Qing Hau Sau III;
10 mg $875   Add to Cart
50 mg $2,000   Add to Cart
64148 Desloratadine Citric Amide
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D64149 Desloratadine Citric Amide-d4
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64153 Desmethoxy Gatifloxacin Trifluoroacetic Acid Salt
10 mg $640   Add to Cart
100 mg $2,120   Add to Cart
9011 (1S,4S)-N-Desmethyl Sertraline HCl
Synonyms:
(1S,4S)- 4-(3,4-Dichlorophenyl)-1,2,3,4-tetrahydro-1- naphthalenamine Hydrochloride;
1 mg $850   Add to Cart
5 mg $1,800   Add to Cart
9012 (1R,4S)-N-Desmethyl Sertraline HCl
Synonyms:
(1R,4S)-4-(3,4-Dichlorophenyl)-1,2,3,4-tetrahydro-1- naphthalenamine Hydrochloride;
1 mg $875   Add to Cart
5 mg $2,000   Add to Cart
9013 (1S,4R)-N-Desmethyl Sertraline HCl
Synonyms:
(1S,4R)-4-(3,4-Dichlorophenyl)-1,2,3,4-tetrahydro-1- naphthalenamine Hydrochloride;
1 mg $875   Add to Cart
5 mg $2,000   Add to Cart
9014 rac-trans-N-Desmethyl Sertraline HCl
Synonyms:
trans-4-(3,4-Dichlorophenyl)-1,2,3,4-tetrahydro-1-naphthalenamine Hydrochloride;
10 mg $845   Add to Cart
50 mg $1,760   Add to Cart
D75238 (±)-cis-N-Desmethylsertraline-1,2,2-d3 Hydrochloride
5 mg $1,000   Add to Cart
25 mg $3,000   Add to Cart
D75239 (±)-trans-N-Desmethylsertraline-1,2,2-d3 Hydrochloride
5 mg $950   Add to Cart
25 mg $2,750   Add to Cart
64217 Dexamethasone 23-Dimorpholinophosphinate
100 mg $625   Add to Cart
250 mg $750   Add to Cart
1 g $1,325   Add to Cart
9324 Didemethylchlorocitalopram
1 mg $860   Add to Cart
5 mg $1,880   Add to Cart
64351 1,2-Dihydro Dexamethasone Phosphate
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64592 α,O-Dimethyl Serotonin HCl
250 mg $640   Add to Cart
2.5 g $2,120   Add to Cart
9594 (E)-1-[4-[2-(N,N-Dimethylamino)ethoxy]phenyl]-1-[4- (trimethylacetoxy)phenyl]-2-phenylbut-1-ene
10 mg $830   Add to Cart
50 mg $1,640   Add to Cart
18045 Epothilone D
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9903 17-Ethoxycarbonyl-6-methoxymorphinan
25 mg $845   Add to Cart
125 mg $1,760   Add to Cart
64967 13-cis-Fenretinide
100 mg $650   Add to Cart
1 g $2,200   Add to Cart
64969 Fenretinide Glucuronide Monosodium Salt
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D64970 Fenretinide Glucuronide Monosodium Salt-d4
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D64966 Fenretinide-d4
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D64968 13-cis-Fenretinide-d4
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65241 3-Hexyl-4-(2-hydroxytridecyl)-2-oxetanone
1 mg $675   Add to Cart
10 mg $2,400   Add to Cart
11037 Z-4-Hydroxy Tamoxifen
Synonyms:
(Z)-4-[1-[4-[2-(Dimethylamino)ethoxy]phenyl]-2-phenyl-1-butenyl] phenol;
10 mg $850   Add to Cart
50 mg $1,800   Add to Cart
10981 (E)-1-(4-Hydroxyphenyl)-1-[4-(trimethylacetoxy)phenyl]-2- phenylbut-1-ene
10 mg $820   Add to Cart
50 mg $1,560   Add to Cart
D65574 Idarubicin-d3
1 mg $2,790   Add to Cart
65575 Idarubicinol (Mixture of Diastereomers)
0.5 mg $675   Add to Cart
5 mg $2,400   Add to Cart
D65576 Idarubicinol-d4 (Mixture of Diastereomers)
0.25 mg $1,475   Add to Cart
1 mg $4,500   Add to Cart
65834 Levophacetoperane
10 mg $650   Add to Cart
100 mg $2,200   Add to Cart
D65835 Levophacetoperane-d3
2.5 mg $650   Add to Cart
25 mg $2,200   Add to Cart
65938 (+)-18-Methoxycoronaridine HCl
10 mg $13,500   Add to Cart
25 mg $17,500   Add to Cart
D65939 (+)-18-Methoxycoronaridine-d4 HCl
5 mg $18,500   Add to Cart
10 mg $20,500   Add to Cart
D65940 (-)-18-Methoxycoronaridine-d4 HCl
5 mg $18,500   Add to Cart
10 mg $20,500   Add to Cart
D66179 2’’-O-Methyl-d3 Paclitaxel
1 mg $700   Add to Cart
10 mg $2,600   Add to Cart
11983 N-Methyl-N-(2-hydroxyethyl)tamoxifen
5 mg $925   Add to Cart
25 mg $2,400   Add to Cart
66339 MT04
10 mg $650   Add to Cart
100 mg $2,200   Add to Cart
65783 Naloxone N-Oxide (100 ug/mL in Acetonitrile)
1 mL $640   Add to Cart
65750 Naloxone N-Oxide (100ug/mL in 1:1 Acetonitrile and water solution )
10 mL $650   Add to Cart
66817 Propoxyphenyl Thiosildenafil
5 mg $650   Add to Cart
50 mg $2,200   Add to Cart
D66818 Propoxyphenyl-thiosildenafil-d8
1 mg $650   Add to Cart
10 mg $2,200   Add to Cart
66849 Prothipendyl HCl
10 mg $650   Add to Cart
100 mg $2,200   Add to Cart
11034 cis-α-Hydroxy Tamoxifen
Synonyms:
(E)-1-[4-[2-(Dimethylamino)ethoxy]phenyl]-1,2-diphenyl-1-butene-3 -ol;
5 mg $835   Add to Cart
25 mg $1,680   Add to Cart
11035 3-Hydroxy Tamoxifen
Synonyms:
3-[(1E)-1-[4-[2-(Dimethylamino)ethoxy]phenyl]-2-phenyl-1-buten-1- yl]-phenol; Droloxifene; E-Droloxifene; K-060; K060E; K 21.060E;
2.5 mg $875   Add to Cart
12.5 mg $2,000   Add to Cart
65524 (Z)-α-Hydroxy Tamoxifen
5 mg $620   Add to Cart
50 mg $1,460   Add to Cart
D65525 (E)-3-Hydroxy Tamoxifen-d5
1 mg $640   Add to Cart
10 mg $2,120   Add to Cart
D11036 3-Hydroxy Tamoxifen-ethyl-d5
Synonyms:
3-[(1E)-1-[4-[2-(Dimethylamino)ethoxy]phenyl]-2-phenyl-1-buten-1- yl-d5]-phenol; Droloxifene-d5; E-Droloxifene-d5; K-060-d5; K060E-d5; K 21.060E-d5;
98%D
1 mg $890   Add to Cart
5 mg $2,120   Add to Cart
D67424 Trityl Olmesartan-d6 Medoxomil
2.5 mg $650   Add to Cart
25 mg $2,200   Add to Cart