Activators

An Activator is a substance that increases the effectiveness of another. For example, a trace quantity of a substance that imparts luminescence to crystals; silver or copper in zinc sulfide or cadmium sulfide pigments. In genetics it would be a molecule that modifies a repressor in a way that enables it to stimulate operon transcription. Examples of activators are: 1-Acetamido-4-cyano-3-methylisoquinoline that is used as a selective inhibitor of cyclic AMP-dependent protein kinase (PKA), while D-erythro-Dihydro-D-sphingosine is used as a Biosynthetic precursor of sphingosine, Inhibits protein kinase C.

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Agonists

Catalog No. Product Name Enrichment
Quantity Price
D39959 trans-Dihydro Lisuride-d10
1 mg $700   Add to Cart
10 mg $2,600   Add to Cart
39938 3-[1-[(1R)-1,2-Dihydro-1-acenaphthylenyl]-4-piperidinyl]-2,3- dihydro-2-oxo-1H-benzimidazole-1-acetic Acid Ethyl Ester
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39978 (E)-1-(2,3-Dihydro-6-methoxy-1H-inden-1-ylidene)-2,3-dihydro-6- methoxy-1H-indene
25 mg $650   Add to Cart
100 mg $950   Add to Cart
250 mg $1,400   Add to Cart
39966 7,8-Dihydroxyflavone
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40009 4’’-Dimethylamino 7,8-Dihydroxyflavone
25 mg $650   Add to Cart
250 mg $2,200   Add to Cart
40008 4’’-Dimethylamino 7,8-Dihydroxyflavone Dimethyl Ether
25 mg $625   Add to Cart
250 mg $2,000   Add to Cart
40010 4-(Dimethylamino)benzoic Acid 6-Acetyl-2,3-dimethoxyphenyl Ester
100 mg $650   Add to Cart
1 g $2,200   Add to Cart
40011 1-[4-(Dimethylamino)phenyl]-3-(2-hydroxy-3,4-dimethoxyphenyl)-1,3 -propanedione
50 mg $650   Add to Cart
500 mg $2,200   Add to Cart
D40013 (8β)-N-[[[3-(Dimethylamino)propyl]amino]carbonyl]-N-ethyl-6- (2-propen-1-yl)-ergoline-8-carboxamide-d5
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39936 (8β)-8-[[[(1,1-Dimethylethyl)dimethylsilyl]oxy]methyl]-6- methylergoline
5 mg $650   Add to Cart
25 mg $950   Add to Cart
100 mg $2,350   Add to Cart
39935 (8β)-8-[[[(1,1-Dimethylethyl)dimethylsilyl]oxy]methyl] ergoline
2.5 mg $625   Add to Cart
10 mg $875   Add to Cart
25 mg $1,250   Add to Cart
40112 2-(3,4-Dimethylphenyl)-1,2-dihydro-5-methyl-3H-pyrazol-3-one
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26421 rac-8-Hydroxy-2-dipropylaminotetralin Hydrobromide
Synonyms:
(±)-8-Hydroxy-2-(dipropylamino)tetralin Hydrobromide; (±)-2-Dipropylamino8-hydroxy-1,2,3,4-tetrahydronaphthalene; (±)-8-Hydroxy-2-(dipropylamino)tetralin; (±)-8-OH-DPAT;
5 mg $860   Add to Cart
50 mg $1,880   Add to Cart
40179 Diquafosol
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40258 Eltrombopag Amide
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40257 Eltrombopag Ethyl Ester
   Request Quote
40259 Eltrombopag Glucuronide
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40256 Eltrombopag Methyl Ester
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40283 (5α)-4,5-Epoxy-14-hydroxy-3-methoxy-6-oxomorphinan-17- carboxylic Acid 1,1-Dimethylethyl Ester
25 mg $650   Add to Cart
250 mg $2,200   Add to Cart
40284 (5α,6β)-4,5-Epoxy-6-[[(2E)-3-(3-furanyl)-1-oxo-2- propenyl]methylamino]-14-hydroxy-3-methoxymorphinan-17-carboxylic Acid 1,1-Dimethylethyl Ester
10 mg $675   Add to Cart
100 mg $2,400   Add to Cart
40286 (5α,6β)-4,5-Epoxy-6-[[(2E)-3-(3-furanyl)-1-oxo-2- propenyl]methylamino]-14-hydroxy-3-methoxymorphinan-17-carboxylic Acid 9H-Fluoren-9-ylmethyl Ester
5 mg $650   Add to Cart
25 mg $1,100   Add to Cart
100 mg $2,775   Add to Cart
40285 (5α,6β)-4,5-Epoxy-6-[[(2E)-3-(3-furanyl)-1-oxo-2- propenyl]methylamino]-3,14-dihydroxymorphinan-17-carboxylic Acid 9H-Fluoren-9-ylmethyl Ester
1 mg $625   Add to Cart
10 mg $2,000   Add to Cart
40290 (8β)-Ergoline-1,6,8-tricarboxylic Acid 1,6-Bis(1,1- dimethylethyl) Ester
0.5 mg $625   Add to Cart
5 mg $2,000   Add to Cart
40289 Ergoline-8β-carboxylic Acid Methyl Ester HCl
0.5 mg $650   Add to Cart
5 mg $2,200   Add to Cart
D40413 Exenatide-d5 Acetate
1 mg $750   Add to Cart
10 mg $3,250   Add to Cart
40418 Fadolmidine HCl
10 mg $650   Add to Cart
100 mg $2,200   Add to Cart
40419 Fadolmidine Methyl Ester
10 mg $625   Add to Cart
100 mg $2,000   Add to Cart
40430 Fedovapagon
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D40431 Fedovapagon-d6
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40444 Fenoldopam
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40445 Fenoldopam HBr
10 mg $640   Add to Cart
100 mg $2,120   Add to Cart
40446 Fenoldopam HCl
   Request Quote
40458 Fexaramine
   Request Quote
D40459 Fexaramine-d4
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40469 Flibanserin HCl
10 mg $610   Add to Cart
25 mg $675   Add to Cart
250 mg $850   Add to Cart
1 g $1,225   Add to Cart
40537 5-Fluoro SDB-005
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40501 1-[[3-Fluoro-4-[5-[(2-fluorophenyl)methyl]-2-benzothiazolyl] phenyl]methyl]-3-azetidinecarboxylic Acid
   Request Quote
40713 Grifolic Acid
   Request Quote
40714 GSA 10
   Request Quote
40715 GSK 1016790A
   Request Quote
40718 GW3965
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40835 (2Z,4E)-5-[(1S)-3-(Hexylthio)-1-hydroxy-2,6,6-trimethyl-4-oxo-2- cyclohexen-1-yl]-3-methyl-2,4-pentadienoic Acid
5 mg $290   Add to Cart
40850 HX 630
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D40851 HX 630-d4
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40900 (8β)-8-(Hydroxymethyl)ergoline-1,6-dicarboxylic Acid 1,6- Bis(1,1-dimethylethyl) Ester
2.5 mg $675   Add to Cart
10 mg $1,025   Add to Cart
25 mg $2,050   Add to Cart
41033 Indacaterol Maleic Acid Salt
1 mg $290   Add to Cart
5 mg $890   Add to Cart
27193 3-Indoxyl Sulfate Potassium Salt
Synonyms:
Indoxyl Sulfate Potassium Salt; Urinary indican; Potassium 3- indoxyl sulfate;
100 mg $900   Add to Cart
1 g $2,700   Add to Cart
D27194 3-Indoxyl Sulfate-d4 Potassium Salt
Synonyms:
1H-Indol-3-ol 3-(Hydrogen Sulfate)-d4 Potassium Salt; 1H-Indol-3-ol Hydrogen Sulfate (Ester)-d4 Monopotassium Salt; Indol-3-yl Potassium Sulfate-d4; Indol-3-ol Potassium Sulfate-d4; Indol-3-yl Sulfate Potassium Salt-d4; Potassium Indol-3-yl Sulfate-d4;
5 mg $1,490   Add to Cart
1 mg $460   Add to Cart
41066 Isoetharine HCl
10 mg $650   Add to Cart
100 mg $2,200   Add to Cart
41068 R,S-Isoetharine HCl
100 mg $625   Add to Cart
250 mg $690   Add to Cart
D41067 Isoetharine-d7 HCl
1 mg $650   Add to Cart
10 mg $2,200   Add to Cart
41114 JWH-180
25 mg $650   Add to Cart
250 mg $2,200   Add to Cart
D41115 JWH-180-d7
1 mg $650   Add to Cart
10 mg $2,200   Add to Cart
41116 JWH-203
25 mg $650   Add to Cart
250 mg $2,200   Add to Cart
D41117 JWH-203-d11
2.5 mg $650   Add to Cart
25 mg $2,200   Add to Cart
41182 Leukadherin 1
10 mg $625   Add to Cart
100 mg $2,000   Add to Cart
41206 Lisuride
0.25 mg $750   Add to Cart
2.5 mg $3,000   Add to Cart
41207 LM 22A4
50 mg $640   Add to Cart
500 mg $2,120   Add to Cart
5 g $2,750   Add to Cart
11392 Lofexidine HCl
Synonyms:
2-[1-(2,6-Dichlorophenoxy)ethyl]-4,5-dihydro-1H-imidazole Hydrochloride; MDL-14042A; Ba-168; Britlofex; Lofetensin; Loxacor;
10 mg $860   Add to Cart
50 mg $1,880   Add to Cart
41215 LY 354740
2.5 mg $650   Add to Cart
25 mg $2,200   Add to Cart
500 mg $9,750   Add to Cart
41216 LY 379268
5 mg $650   Add to Cart
10 mg $750   Add to Cart
50 mg $2,150   Add to Cart
41217 LY 456236
10 mg $610   Add to Cart
50 mg $940   Add to Cart
100 mg $1,250   Add to Cart
41242 MCOPPB TriHCl
10 mg $675   Add to Cart
100 mg $2,400   Add to Cart
41303 Methoxamine HCl (Mixture of Diastereomers)
250 mg $650   Add to Cart
2.5 g $2,200   Add to Cart
41307 1-(4’’-Methoxy[1,1’’-biphenyl]-2-yl)-piperazine HCl
10 mg $640   Add to Cart
100 mg $2,120   Add to Cart
41442 N-Methyl Fenoldopam HCl
2.5 mg $610   Add to Cart
10 mg $830   Add to Cart
25 mg $1,125   Add to Cart
41374 2,2’’-(Methylazanediyl)bis(1-(3-hydroxyphenyl)ethanone) HCl
25 mg $625   Add to Cart
100 mg $875   Add to Cart
250 mg $1,250   Add to Cart
41650 ML-179
10 mg $650   Add to Cart
25 mg $800   Add to Cart
100 mg $2,050   Add to Cart
41653 ML-233
10 mg $650   Add to Cart
50 mg $1,075   Add to Cart
100 mg $2,025   Add to Cart
41651 ML-335
10 mg $650   Add to Cart
50 mg $1,075   Add to Cart
100 mg $2,025   Add to Cart
41670 Mosapride
10 mg $610   Add to Cart
100 mg $1,380   Add to Cart
41669 Mosapride Citrate Dihydrate
10 mg $610   Add to Cart
50 mg $875   Add to Cart
250 mg $1,475   Add to Cart
1 g $2,475   Add to Cart
12405 Mosapride citrate salt dihydrate
Synonyms:
4-amino-5-chloro-2-ethoxy-N-[[4-(4-fluorophenyl)methyl]-2- morpholinyl]methyl]-benzamide;
10 mg $860   Add to Cart
50 mg $1,880   Add to Cart
12413 Muraglitazar
Synonyms:
N-[(4-Methoxyphenoxy)carbonyl]-N-[[4-[2-(5-methyl-2-phenyl-4- oxazolyl)ethoxy]phenyl]methyl]glycine; BMS 298585; Pargluva;
1 mg $990   Add to Cart
5 mg $2,120   Add to Cart
10 mg $2,900   Add to Cart
D41682 Nalfurafine N-Oxide-d3
1 mg $680   Add to Cart
10 mg $2,440   Add to Cart
13446 1-Hydroxy-2-naphthoate-Salmeterol
Synonyms:
Salmeterol xinafoate; GR-33343G; Arial; Salmetedur; Serevent;
10 mg $875   Add to Cart
50 mg $2,000   Add to Cart
41689 NDT 9513727
10 mg $680   Add to Cart
50 mg $1,350   Add to Cart
100 mg $2,440   Add to Cart
D41690 NDT 9513727-d9
2.5 mg $650   Add to Cart
25 mg $2,200   Add to Cart
41705 9-Nitro Oleic Acid
5 mg $650   Add to Cart
50 mg $2,200   Add to Cart
41764 NS 3623
10 mg $650   Add to Cart
50 mg $1,150   Add to Cart
100 mg $2,050   Add to Cart
41766 O-1602
5 mg $610   Add to Cart
10 mg $625   Add to Cart
25 mg $725   Add to Cart
41887 PD-149163
10 mg $660   Add to Cart
100 mg $2,280   Add to Cart
41979 L-Phenylalanyl-L-seryl-L-leucyl-L-leucyl-L-arginyl-L-tyrosinamide
2.5 mg $650   Add to Cart
5 mg $675   Add to Cart
25 mg $1,250   Add to Cart
D41987 Phenylephrine-d3 hydrochloride (methyl-d3)
1 mg $590   Add to Cart
5 mg $1,490   Add to Cart
14847 Pimavanserin
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30386 Pregnenolone Acetate
Synonyms:
3β-Acetoxy-5-pregnen-20-one; 5-Pregnen-3β-ol-20-one Acetate;
25 mg $900   Add to Cart
250 mg $2,700   Add to Cart
42081 Promethazine Sulfone
2.5 mg $675   Add to Cart
25 mg $1,275   Add to Cart
100 mg $2,400   Add to Cart
42122 PSB-SB1202
2.5 mg $650   Add to Cart
10 mg $950   Add to Cart
25 mg $1,400   Add to Cart
D32505 (+/-)-Ractopamine-d3 hydrochloride 97%D
5 mg $690   Add to Cart
13340 rac Ramelteon
Synonyms:
rac N-[-[(8S)-1,6,7,8-Tetrahydro-2H-indeno[5,4-β]furan-8-yl] ethyl]propanamide; rac Rozerem;
2.5 mg $875   Add to Cart
12.5 mg $2,000   Add to Cart
D75066 Ramelteon-d5
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D13342 rac Ramelteon-d3
Synonyms:
rac N-[[1,6,7,8-Tetrahydro-2H-indeno[5,4-β]furan-8-yl]ethyl] propanamide-d3; rac TAK-375-d3; rac Rozerem-d3; 		98%D
1 mg $925   Add to Cart
5 mg $2,400   Add to Cart
13361 Regadenoson
Synonyms:
2-[4-[(Methylamino)carbonyl]-1H-pyrazol-1-yl]-adenosine;
5 mg $900   Add to Cart
25 mg $2,200   Add to Cart
42166 Resiquimod
10 mg $490   Add to Cart
42174 Rilmenidine Phosphate
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42175 Rimiterol HBr
10 mg $650   Add to Cart
100 mg $2,200   Add to Cart
D42176 Rimiterol-d4 HBr
2.5 mg $650   Add to Cart
25 mg $2,200   Add to Cart
13405 Rimonabant hydrochloride
Synonyms:
Acomplia, SR141716;
10 mg $190   Add to Cart
50 mg $590   Add to Cart
18761 Ritodrine HCl
5 mg $950   Add to Cart
25 mg $1,500   Add to Cart
42180 Rizatriptan Bismethylammonium Chloride Dimer
10 mg $675   Add to Cart
100 mg $2,400   Add to Cart
D4398 Rizatriptan-d6 Benzoate
Synonyms:
(N,N-Dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-1H-indole-3- ethanamine-D6); 		98%D
1 mg $750   Add to Cart
5 mg $1,995   Add to Cart
42181 RO 5256390
Synonyms:
(S)-4-((S)-2-Phenylbutyl)-4,5-dihydrooxazol-2-amine;
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CD42182 RO 5256390-13C, d2
1 mg $685   Add to Cart
10 mg $2,440   Add to Cart
13436 Rotigotine HCl
Synonyms:
(6S)-5,6,7,8-Tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-1- naphthalenol; (-)-N 0437; N 0923; Neupro; SPM 962;
5 mg $925   Add to Cart
25 mg $2,400   Add to Cart
D13437 rac Rotigotine-d3
Synonyms:
(6S)-5,6,7,8-Tetrahydro-6-[propyl-d3[2-(2-thienyl)ethyl]amino ]-1-naphthalenol; (-)-N 0437-d3; N 0923-d3; Neupro-d3; Rotigotine-d3; SPM 962-d3; 		98%D
1 mg $925   Add to Cart
5 mg $2,400   Add to Cart
42188 RWJ-52353 HCl
10 mg $640   Add to Cart
100 mg $2,120   Add to Cart
18767 Salmeterol
Synonyms:
(RS)-2-(hydroxymethyl)-4-[1-hydroxy-2-[6-(4-phenylbutoxy) hexylamino]ethyl]phenol;
10 mg $290   Add to Cart
42193 Salvinorin B
2.5 mg $650   Add to Cart
25 mg $2,200   Add to Cart
42199 SB 334867
10 mg $650   Add to Cart
100 mg $2,200   Add to Cart
38455 N-Acetyl-SB-611855 Glucuronide Disodium Salt
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42211 Sipoglitazar
5 mg $675   Add to Cart
50 mg $2,400   Add to Cart
42214 SKF 38393 HCl
100 mg $625   Add to Cart
250 mg $675   Add to Cart
2.5 g $2,400   Add to Cart
C42215 SKF 81297C
10 mg $615   Add to Cart
25 mg $675   Add to Cart
100 mg $1,050   Add to Cart
42252 SR 1078
10 mg $610   Add to Cart
110 mg $1,380   Add to Cart
D32421 Succinyl(choline-1,1,1’,1’,2,2,2’,2’-d8) Bromide 99%D
50 mg $590   Add to Cart
D3131 Succinylcholine Chloride-d8 98%D
50 mg $590   Add to Cart
42273 Sumatriptan Hydroxy-Oxindole Impurity (Sumatriptan Impurity 1)
0.5 mg $725   Add to Cart
5 mg $2,975   Add to Cart
13620 Sumatriptan Succinate
Synonyms:
3-[2-(Dimethylamino)ethyl]-N-methyl-1H-indole-5- methanesulfonamide, Succinate, Imigran, Imitrex,; 1-(3-(2-(Dimethylamino)ethyl)-1H-indol-5-yl)-N- methylmethanesulfonamide succinate;
50 mg $860   Add to Cart
250 mg $1,880   Add to Cart
D13621 Sumatriptan-d6 Succinate
Synonyms:
3-[2-(Dimethyl-d6-amino)ethyl]-N-methyl-1H-indole-5- methanesulfonamide, Succinate, Imigran, Imitrex,; 		98%D
1 mg $875   Add to Cart
5 mg $2,000   Add to Cart
D75224 Sumatriptan-d6 Hemisuccinate
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18786 Talipexole DiHCl
5 mg $950   Add to Cart
25 mg $1,500   Add to Cart
42295 Telmisartan Impurity B
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42349 3α,5α-Tetrahydronorethisterone
2.5 mg $650   Add to Cart
25 mg $2,200   Add to Cart
42351 3β,5α-Tetrahydronorethisterone
10 mg $650   Add to Cart
100 mg $2,200   Add to Cart
D42350 3α,5α-Tetrahydronorethisterone-d5
10 mg $2,600   Add to Cart
D42352 3β,5α-Tetrahydronorethisterone-d5
10 mg $2,600   Add to Cart
C39516 2C-TFM HCl
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D13807 Thiomuscimol-d3 98%D
1 mg $875   Add to Cart
5 mg $2,000   Add to Cart
42405 Tiospirone HCl
10 mg $650   Add to Cart
100 mg $2,200   Add to Cart
D42406 Tiospirone-d8 HCl
1 mg $650   Add to Cart
10 mg $2,200   Add to Cart
13844 Tizanidine hydrochloride
Synonyms:
5-Chloro-N-(4,5-dihydro-1H-imidazol-2-yl)-2,1,3-benzothiadiazol-4 -amine hydrochloride; AB-021; DS-103-282; Sirdalud; Ternelin; Zanaflex;
1 g $490   Add to Cart
5 g $1,425   Add to Cart
D3732 Tizanidine-d4 98%D
1 mg $390   Add to Cart
D3855 N-Acetyl Tizanidine-d4
Synonyms:
1-[2-[(5-Chloro-2,1,3-benzothiadiazol-4-yl)amino]-4,5-dihydro-1H- imidazol-1-yl-D4]-ethanone; 		98%D
1 mg $650   Add to Cart
5 mg $1,800   Add to Cart
42509 7,8,3’’-Trihydroxyflavone
100 mg $640   Add to Cart
1 g $2,120   Add to Cart
14105 Tulobuterol
Synonyms:
2-Chloro-α-[[(1,1-dimethylethyl)amino]methyl]benzenemethanol;
100 mg $870   Add to Cart
0.5 g $1,960   Add to Cart
42622 W 212393
2.5 mg $675   Add to Cart
25 mg $2,400   Add to Cart
42626 WIN 54461
5 mg $725   Add to Cart
50 mg $2,500   Add to Cart
42625 Win 55212-2
25 mg $7,250   Add to Cart
42627 Xamoterol
10 mg $650   Add to Cart
100 mg $2,200   Add to Cart
D42628 Xamoterol-d5
1 mg $650   Add to Cart
10 mg $2,200   Add to Cart
14846 Zamifenacin
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14692 Zilpaterol HCl
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42635 ZK-994
10 mg $28,500   Add to Cart
D14220 Zolmitriptan-d6 (Major) N-Oxide
Synonyms:
(4S)-4-[[3-[2-(Dimethyl-d6-oxidoamino)ethyl]-1H-indol-5-yl] methyl-2-oxazolidinone;
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