Product:
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MDV3100 ( Enzalutamide ) |
Catalog Number:
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111366 |
CAS Number:
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915087-33-1 |
Synonyms:
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Enzalutamide, MDV3100, MDV-3100, MDV 3100; Chemical Name: 4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluoro-N-methylbenzamide |
Pricing:
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Formula:
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C21H16F4N4O2S |
Molecular Weight:
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464.4 |
Structure:
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Appearance:
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Solid |
Category:
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Nucleotides and Nucleosides Alphabetic Listing |
Solubility:
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≥23.22 mg/mL in DMSO; insoluble in H2O; ≥9.44 mg/mL in EtOH |
Transportation:
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Ships on blue ice |
Literature References:
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Manoj P. Menon, Celestia S. Higano. Enzalutamide, a Second Generation Androgen Receptor Antagonist: Development and Clinical Applications in Prostate Cancer. Current Oncology Reports. 2013; 15(2): 69–75. |
MSDS:
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Applications:
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MDV3100, known as Enzalutamide, is a second-generation androgen receptor (AR) signaling inhibitor. It has been demonstrated impressive affinity to the AR compared to the first-generation AR inhibitors. |